Journal
ORGANIC LETTERS
Volume 14, Issue 3, Pages 836-839Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol203360g
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Funding
- Japan Private School Promotion Foundation
- MEXT
- Grants-in-Aid for Scientific Research [24590025, 23710261] Funding Source: KAKEN
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A novel copper-catalyzed [5 + 1] annulation of 2-ethynylanilines with an N,O-acetal, which functioned as a Cl part, leading to the preparation of quinoline derivatives with an ester substituent on the 2-position is described. A combination of CuBr2 and trifluoroacetic acid (TFA) promoting [5 + 1] annulation of the 2-ethynylaniline with ethyl glyoxylate is also demonstrated.
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