Journal
ORGANIC LETTERS
Volume 14, Issue 2, Pages 664-667Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol203392r
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Funding
- MEXT
- JSPS, Japan
- Grants-in-Aid for Scientific Research [22750040] Funding Source: KAKEN
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A wide range of o-alkynylanilines undergo a copper-catalyzed direct C-H/N-H coupling with azoles followed by benzannulation to form the corresponding N-azolylindoles in good yields. The domino reaction proceeds effectively with molecular oxygen as the sole oxidant and provides a new dehydrogenative access to the titled compounds of interest in pharmaceutical and material sciences.
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