Journal
ORGANIC LETTERS
Volume 12, Issue 14, Pages 3168-3171Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol101078z
Keywords
-
Categories
Funding
- National Sciences and Engineering Research Counsil of Canada
- Egyptian Academy of Scientific Research and Technology
Ask authors/readers for more resources
A new method for the synthesis of 5-azaindole derivatives is reported. A [3+2] dipolar cycloaddition between nitriles and a 3,4-cyclopropanopiperidirie followed by SeO2 oxidation affords the target compounds in moderate to excellent yields. The divergent nature and cost effectiveness of this method makes it very suitable for combinatorial applications in the pharmaceutical industry.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available
Share Paper
