Journal
ORGANIC LETTERS
Volume 11, Issue 8, Pages 1677-1680Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol802882k
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- CDTI (Spanish Ministry of Research and Science)
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N-Methylanilines are readily synthesized in high yields through the copper(II)-promoted coupling of anilines and methylboronic acid. This method represents a new approach for the selective monomethylation of anilines, and it is the first reported example of a Chan-Lam coupling involving the use of methylboronic acid. An incubation period of the substrate with the copper reagent is needed before addition of the methylboronic acid.
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