Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 12, Issue 31, Pages 5822-5826Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c4ob01019a
Keywords
-
Categories
Funding
- Okinawa Institute of Science and Technology Graduate University
- MEXT (Japan)
- Grants-in-Aid for Scientific Research [24105535, 26105757] Funding Source: KAKEN
Ask authors/readers for more resources
One-pot syntheses of polysubstituted 3-acylpyrroles from readily available unsaturated ketones and N-substituted propargylated amines have been developed. An aza-Michael/alkyne carbocyclization cascade, by cooperative catalysis using pyrrolidine and a copper salt, followed by oxidation in situ gave 3-acylpyrroles, which were also transformed further to functionalized, highly substituted 3-acylpyrroles.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available