Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 11, Issue 38, Pages 6470-6476Publisher
ROYAL SOC CHEMISTRY
DOI: 10.1039/c3ob41349g
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Funding
- CONACYT [CB-2011-166747-Q, CVU 176745, 290662_UG, 290735_UG, 209265/229559, 230777/209054, 368973/250842, CB-2011-168474]
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A series of nine novel 3-tetrazolylmethyl-azepino[4,5-b]indol-4-ones were prepared in moderate to good overall yields in only two reaction steps. The first step consisted of a one-pot sequential process of an Ugi-azide multicomponent reaction, N-acylation and S(N)2 to give the xanthates. The second step was an intramolecular cyclization under free radical conditions. Also, their binding modes have been modelled using docking techniques.
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