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RS Muthyala et al.
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Synthesis, binding affinity, and transcriptional activity of hydroxy- and methoxy-substituted 3,4-diarylsalicylaldoximes on estrogen receptors α and β
F Minutolo et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 2. Clinical considerations and new agents
VC Jordan
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions
VC Jordan
JOURNAL OF MEDICINAL CHEMISTRY (2003)
Estrogenic diazenes: Heterocyclic non-steroidal Estrogens of unusual structure with selectivity for estrogen receptor subtypes
U Ghosh et al.
BIOORGANIC & MEDICINAL CHEMISTRY (2003)
2-phenylspiroindenes: A novel class of Selective Estrogen Receptor Modulators (SERMs)
TA Blizzard et al.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2003)
Molecular basis for the subtype discrimination of the estrogen receptor-β-selective ligand diarylpropionitrile
J Sun et al.
MOLECULAR ENDOCRINOLOGY (2003)
Advances in the science of estrogen receptor modulation
MJ Meegan et al.
CURRENT MEDICINAL CHEMISTRY (2003)
Estrogen receptor (ER)-β reduces ERα-regulated gene transcription, supporting a Ying Yang relationship between ERα and ERβ in mice
MK Lindberg et al.
MOLECULAR ENDOCRINOLOGY (2003)
Differential expression of the estrogen receptor beta (ERβ) in human prostate tissue, premalignant changes, and in primary, metastatic, and recurrent prostatic adenocarcinoma
T Fixemer et al.
PROSTATE (2003)
Declining estrogen receptor-beta expression defines malignant progression of human breast neoplasia
AM Shaaban et al.
AMERICAN JOURNAL OF SURGICAL PATHOLOGY (2003)
A new series of estrogen receptor modulators that display selectivity for estrogen receptor β
BR Henke et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Effect of ovariectomy on adipose tissue of mice in the absence of estrogen receptor alpha (ERα):: a potential role for estrogen receptor beta (ERβ)
A Naaz et al.
HORMONE AND METABOLIC RESEARCH (2002)
Characterization of the biological roles of the estrogen receptors, ERα and ERβ, in estrogen target tissues in vivo through the use of an ERα-selective ligand
HA Harris et al.
ENDOCRINOLOGY (2002)
Oestrogen receptor β in breast cancer:: good, bad or still too early to tell?
V Speirs
JOURNAL OF PATHOLOGY (2002)
Toward selective ERβ Agonists for central nervous system disorders:: Synthesis and characterization of aryl benzthiophenes
U Schopfer et al.
JOURNAL OF MEDICINAL CHEMISTRY (2002)
Abnormal vascular function and hypertension in mice deficient in estrogen receptor β
Y Zhu et al.
SCIENCE (2002)
Estrogen receptor-β potency-selective ligands:: Structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues
MJ Meyers et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
Salicylaldoxime moiety as a phenolic A-ring substitute in estrogen receptor ligands
F Minutolo et al.
JOURNAL OF MEDICINAL CHEMISTRY (2001)
Increased anxiety and synaptic plasticity in estrogen receptor β-deficient mice
W Krezel et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)
The role of estrogen and estrogen receptor-α in male adipose tissue
PS Cooke et al.
MOLECULAR AND CELLULAR ENDOCRINOLOGY (2001)
Estrogen receptors α and β in the normal, hyperplastic and carcinomatous human prostate
M Royuela et al.
JOURNAL OF ENDOCRINOLOGY (2001)
Estrogen receptor α, not β, is a critical link in estradiol-mediated protection against brain injury
DB Dubal et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2001)
Role of estrogen receptor beta in estrogen action
K Pettersson et al.
ANNUAL REVIEW OF PHYSIOLOGY (2001)
Pyrazole ligands:: Structure-affinity/activity relationships and estrogen receptor-α-selective agonists
SR Stauffer et al.
JOURNAL OF MEDICINAL CHEMISTRY (2000)
Increased adipose tissue in male and female estrogen receptor-α knockout mice
PA Heine et al.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (2000)
Immunolocalisation of oestrogen receptor beta in human tissues
AH Taylor et al.
JOURNAL OF MOLECULAR ENDOCRINOLOGY (2000)