4.2 Article

Three-dimensional quantitative structure-activity relationship CoMFA/CoMSIA on pyrrolidine-based tartrate diamides as TACE inhibitors

Related references

Note: Only part of the references are listed.
Article Biochemistry & Molecular Biology

3D-QSAR Studies of JNK1 Inhibitors Utilizing Various Alignment Methods

Thirumurthy Madhavan et al.

CHEMICAL BIOLOGY & DRUG DESIGN (2012)

Article Chemistry, Medicinal

2-(2-Aminothiazol-4-yl)pyrrolidine-based tartrate diamides as potent, selective and orally bioavailable TACE inhibitors

Chaoyang Dai et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2011)

Article Chemistry, Medicinal

Synthesis, preliminary biological evaluation and molecular modeling of some new heterocyclic inhibitors of TACE

Prabal Sengupta et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2011)

Article Chemistry, Multidisciplinary

Open Babel: An open chemical toolbox

Noel M. O'Boyle et al.

JOURNAL OF CHEMINFORMATICS (2011)

Article Chemistry, Medicinal

Structure and activity relationships of tartrate-based TACE inhibitors

Dansu Li et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)

Article Chemistry, Medicinal

The discovery of novel tartrate-based TNF-α converting enzyme (TACE) inhibitors

Kristin E. Rosner et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2010)

Article Chemistry, Medicinal

3D-QSAR analysis of human immunodeficiency virus entry-1 inhibitors by CoMFA and CoMSIA

Somayeh Pirhadi et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)

Article Chemistry, Medicinal

3D-QSAR studies on quinazoline antifolate thymidylate synthase inhibitors by CoMFA and CoMSIA models

Vivek Srivastava et al.

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (2010)

Review Chemistry, Medicinal

Novel TACE inhibitors in drug discovery: a review of patented compounds

Prashant R. Murumkar et al.

EXPERT OPINION ON THERAPEUTIC PATENTS (2010)

Review Pharmacology & Pharmacy

TNF alpha in atherosclerosis, myocardial ischemia/reperfusion and heart failure

Petra Kleinbongard et al.

PHARMACOLOGY & THERAPEUTICS (2010)

Review Biochemistry & Molecular Biology

Current perspective of TACE inhibitors: A review

Shirshendu DasGupta et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2009)

Article Biochemistry & Molecular Biology

Synthesis and activity of tryptophan sulfonamide derivatives as novel non-hydroxamate TNF-α converting enzyme (TACE) inhibitors

Kaapjoo Park et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2009)

Article Biochemistry & Molecular Biology

Chromen-based TNF-alpha converting enzyme (TACE) inhibitors: Design, synthesis, and biological evaluation

Kwangwoo Chun et al.

BIOORGANIC & MEDICINAL CHEMISTRY (2008)

Article Chemistry, Organic

Novel thiol-based TACE inhibitors. Part 2: Rational design, synthesis, and SAR of thiol-containing aryl sulfones

Upul K. Bandarage et al.

BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (2007)