Journal
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
Volume 132, Issue 38, Pages 13194-13196Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ja1066459
Keywords
-
Categories
Funding
- NIH/NIGMS [GM-073949]
- NSF
- Japan Society for the Promotion of Science (JSPS)
- Amgen
- Bristol-Myers Squibb
Ask authors/readers for more resources
A direct arylation of a variety of electron-deficient heterocycles with arylboronic acids has been developed. This new reaction proceeds readily at room temperature using inexpensive reagents: catalytic silver(I) nitrate in the presence of persulfate cooxidant. The scope with respect to heterocycle and boronic acid coupling partner is broad, and sensitive functional groups are tolerated. This method allows for rapid access to a variety of arylated heterocycles that would be more difficult to access with traditional methods.
Authors
I am an author on this paper
Click your name to claim this paper and add it to your profile.
Reviews
Recommended
No Data Available