Journal
JOURNAL OF ORGANIC CHEMISTRY
Volume 74, Issue 15, Pages 5675-5678Publisher
AMER CHEMICAL SOC
DOI: 10.1021/jo900752z
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Funding
- Korea Science and Engineering Foundation (KOSEF) [R15-2003-012-02001-0]
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TBAF-assisted N-arylation and benzylation of benzazoles such as I H-benzimidazole, 1H-indole, and 1H-benzotriazole with aryl and benzyl halides have been demonstrated tinder the ligand/base/solvent-free conditions. In the presence of CuBr2 and TBAF (n-Bu4NF), the azoles underwent N-arylation and benzylation with aryl and benzyl halides smoothly in moderate to good yields. It is noteworthy that the reaction is conducted under the ligand/base/solvent-free conditions.
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