Journal
ORGANIC LETTERS
Volume 17, Issue 18, Pages 4588-4591Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.5b02320
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Funding
- Max-Planck-Gesellschaft
- Council on Grants of the President of the Russian Federation (Program for State Support of Leading Scientific Schools) [NSh-3656.2014.3]
- Russian Foundation for Basic Research [13-03-01271]
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A novel, mild, and practical method of amination of simple nonfunctionalized arenes under metal free conditions has been developed. The approach allows coupling of electron-rich arenes with amino derivatives of electron-deficient heterocycles providing rapid access to scaffolds of bioactive compounds and is based on the application of the hypervalent iodine(III) reagent as an oxidant. Regioselective functionalization of C-H bonds of arenes by the formation of C-N bonds under organocatalytic conditions was demonstrated.
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