Journal
ORGANIC LETTERS
Volume 17, Issue 3, Pages 664-667Publisher
AMER CHEMICAL SOC
DOI: 10.1021/ol503689r
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- Chinese Scholarship Council
- Deutsche Forschungsgemeinschaft (DFG)
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Diastereoselective oxyarylation of N-protected 2-alkylindoles with commercially available boronic acids and TEMPO as a mild oxidant to give N-protected 2-aryl-2-alkyl-3-(2-chloroacetoxy)indolines is described. Reactions are easy to conduct, and product indolines containing a fully substituted C-center are obtained in good yields with good to excellent selectivities.
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