Journal
ORGANIC LETTERS
Volume 17, Issue 16, Pages 4014-4017Publisher
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.5b01909
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Funding
- National Natural Science Foundation of China [21121062, 21432011, 21272250]
- National Basic Research Program of China (973 Program) [2015CB856600]
- Chinese Academy of Sciences
- National Science Foundation [CHE-1152767, CHE-1465106]
- National Institutes of Health [R01-GM098777]
- Division Of Chemistry
- Direct For Mathematical & Physical Scien [1624216] Funding Source: National Science Foundation
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A one-pot asymmetric synthesis of 1,2,3,4-tetrahydrocarbizoles has been developed via an enantioselective [3 + 3] annulation of 2-alkynylindoles and donor acceptor cyclopropanes. In the presence of chiral Lewis acids as catalysts, a series of optically active tetrahydrocarbazoles were furnished in high yields (63-87%) With good to excellent levels of enantioselectivity (up to 94% ee).
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