4.8 Article

The ins and outs of selective kinase inhibitor development

Related references

Note: Only part of the references are listed.
Review Biochemistry & Molecular Biology

Exploration of Type II Binding Mode: A Privileged Approach for Kinase Inhibitor Focused Drug Discovery?

Zheng Zhao et al.

ACS CHEMICAL BIOLOGY (2014)

Article Pharmacology & Pharmacy

Recently targeted kinases and their inhibitors - the path to clinical trials

Stefan Knapp et al.

CURRENT OPINION IN PHARMACOLOGY (2014)

Article Biochemistry & Molecular Biology

A unique inhibitor binding site in ERK1/2 is associated with slow binding kinetics

Apirat Chaikuad et al.

NATURE CHEMICAL BIOLOGY (2014)

Article Biochemistry & Molecular Biology

Dual kinase-bromodomain inhibitors for rationally designed polypharmacology

Pietro Ciceri et al.

NATURE CHEMICAL BIOLOGY (2014)

Article Medicine, General & Internal

Resistance Mechanisms for the Bruton's Tyrosine Kinase Inhibitor Ibrutinib

Jennifer A. Woyach et al.

NEW ENGLAND JOURNAL OF MEDICINE (2014)

Review Biochemistry & Molecular Biology

Developing Irreversible Inhibitors of the Protein Kinase Cysteinome

Qingsong Liu et al.

CHEMISTRY & BIOLOGY (2013)

Article Ophthalmology

Topical Antiangiogenic SRPK1 Inhibitors Reduce Choroidal Neovascularization in Rodent Models of Exudative AMD

Melissa V. Gammons et al.

INVESTIGATIVE OPHTHALMOLOGY & VISUAL SCIENCE (2013)

Article Biochemistry & Molecular Biology

Targeting Diverse Signaling Interaction Sites Allows the Rapid Generation of Bivalent Kinase Inhibitors

Zachary B. Hill et al.

ACS CHEMICAL BIOLOGY (2012)

Article Biochemistry & Molecular Biology

Skepinone-L is a selective p38 mitogen-activated protein kinase inhibitor

Solveigh C. Koeberle et al.

NATURE CHEMICAL BIOLOGY (2012)

Article Chemistry, Medicinal

Understanding the Impact of the P-loop Conformation on Kinase Selectivity

Cristiano R. W. Guimaraes et al.

JOURNAL OF CHEMICAL INFORMATION AND MODELING (2011)

Article Biotechnology & Applied Microbiology

Comprehensive analysis of kinase inhibitor selectivity

Mindy I. Davis et al.

NATURE BIOTECHNOLOGY (2011)

Article Biochemistry & Molecular Biology

Specific Btk inhibition suppresses B cell- and myeloid cell-mediated arthritis

Julie A. Di Paolo et al.

NATURE CHEMICAL BIOLOGY (2011)

Article Multidisciplinary Sciences

Targeting Bcr-Abl by combining allosteric with ATP-binding-site inhibitors

Jianming Zhang et al.

NATURE (2010)

Article Biochemistry & Molecular Biology

The (un)targeted cancer kinome

Oleg Fedorov et al.

NATURE CHEMICAL BIOLOGY (2010)

Article Biochemistry & Molecular Biology

Structure and allosteric effects of low-molecular-weight activators on the protein kinase PDK1

Valerie Hindie et al.

NATURE CHEMICAL BIOLOGY (2009)

Article Biochemistry & Molecular Biology

Activation segment dimerization: a mechanism for kinase autophosphorylation of non-consensus sites

Ashley C. W. Pike et al.

EMBO JOURNAL (2008)

Article Biotechnology & Applied Microbiology

Quantitative chemical proteomics reveals mechanisms of action of clinical ABL kinase inhibitors

Marcus Bantscheff et al.

NATURE BIOTECHNOLOGY (2007)

Article Chemistry, Multidisciplinary

Ruthenium half-sandwich complexes bound to protein kinase Pim-1

JE Debreczeni et al.

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION (2006)

Article Biotechnology & Applied Microbiology

A small molecule-kinase interaction map for clinical kinase inhibitors

MA Fabian et al.

NATURE BIOTECHNOLOGY (2005)

Article Multidisciplinary Sciences

Structural mechanism for STI-571 inhibition of Abelson tyrosine kinase

T Schindler et al.

SCIENCE (2000)